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We have discovered that 17beta- N,N- diethyl carbamoyl -6-azaandrost-4-en-3-one is a time-dependent inhibitor of type II 5alpha-reductase, as is the drug finasteride, anabola testosteron methenolone enanthate. To 10 mg of Tren dissolved in 10 mL of anhydrous THF, 100 ?L of potassium tri-sec-butylborohydride 1 M in THF were added under constant stirring. After 15 min, the reaction was stopped with 10 mL of ultrapure water, and subsequently, a LLE with 20 mL of TBME was performed. An aliquot of the yielded products was acetylated as described in section Acetylation, . Metabolite Identification With GC-TC-IRMS..
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